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G Protein-selective GPCR Conformations Measured Using FRET Sensors in a Live Cell Suspension Fluorometer Assay
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The use of conformationally thermostabilised GPCRs in drug discovery: application to fragment, structure and

Benjamin G Tehan1, John A Christopher1

  • 1Heptares Therapeutics, Biopark, Broadwater Road, Welwyn Garden City, Hertfordshire AL7 3AX, United Kingdom.

Current Opinion in Pharmacology
|July 12, 2016
PubMed

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