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Updated: Mar 17, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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Potential for the Rational Design of Allosteric Modulators of Class C GPCRs

John A Christopher1, Andrew S Doré, Benjamin G Tehan

  • 1Heptares Therapeutics Ltd., Biopark, Welwyn Garden City, Hertfordshire, U.K. john.christopher@heptares.com.

Current Topics in Medicinal Chemistry
|July 25, 2016
PubMed

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