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Binding characterization, synthesis and biological evaluation of RXRα antagonists targeting the coactivator binding

Dingyu Xu1, Shangjie Guo1, Ziwen Chen1

  • 1School of Pharmaceutical Sciences, Xiamen University, Xiamen 361005, China.

Bioorganic & Medicinal Chemistry Letters
|July 25, 2016
PubMed

Keywords:
Coactivator-binding site ligandCoregulator-binding siteNuclear receptorsRXRα modulatorsTNFα/NF-κB pathway

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