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Design and evaluation of 1,7-naphthyridones as novel KDM5 inhibitors

Sharada S Labadie1, Peter S Dragovich1, Richard T Cummings2

  • 1Genentech Inc., 1 DNA Way, South San Francisco, CA 94080, USA.

Bioorganic & Medicinal Chemistry Letters
|August 9, 2016
PubMed

Keywords:
EpigeneticsHistone lysine demethylasesKDM5 inhibitors

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