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Identification of acylthiourea derivatives as potent Plk1 PBD inhibitors

Taikangxiang Yun1, Tan Qin2, Ying Liu3

  • 1Center for Quantitative Biology, Academy for Advanced Interdisciplinary Studies, Peking University, Beijing 100871, China.

European Journal of Medicinal Chemistry
|September 5, 2016
PubMed

Keywords:
Binding affinityHalogenosulfamoylphenyl acylthioureaIn vitro assayPolo-box domainPolo-like kinase 1Small molecular inhibitor

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