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4,5-Disubstituted 6-Aryloxy-1,3-dihydrobenzo[c][1,2]oxaboroles Are Broad-Spectrum Serine β-Lactamase Inhibitors

David C McKinney1, Fei Zhou1, Charles J Eyermann1

  • 1Infection Innovative Medicines, AstraZeneca R&D Boston , 35 Gatehouse Drive, Waltham Massachusetts 02451, United States.

ACS Infectious Diseases
|September 14, 2016
PubMed

Keywords:
Gram-negative infectionsoxaborolesstructure-guided designβ-lactamase inhibitors

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