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Method for Identifying Small Molecule Inhibitors of the Protein-protein Interaction Between HCN1 and TRIP8b
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Tetrahydroindazole derivatives as potent and peripherally selective cannabinoid-1 (CB1) receptor inverse agonists

Jay M Matthews1, James J McNally1, Peter J Connolly1

  • 1Janssen Research & Development, L.L.C., Welsh & McKean Roads, Spring House, PA 19477, USA(†).

Bioorganic & Medicinal Chemistry Letters
|September 28, 2016
PubMed

Keywords:
CB1 receptorCannabinoid receptorInverse agonistPeripheral selectivityPeripherally restricted

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