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Palladium-Catalyzed Arylation of Carbasugars Enables the Discovery of Potent and Selective SGLT2 Inhibitors

Wai-Lung Ng1,2, Kit-Man Lau3, Clara B-S Lau3

  • 1Department of Chemistry, The Chinese University of Hong Kong, Shatin, New Territories, Hong Kong SAR, China.

Angewandte Chemie (International Ed. in English)
|October 5, 2016
PubMed

Keywords:
carbohydratescross-couplingdrug designinhibitorspalladium

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