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Updated: Mar 13, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Synthesis and biological evaluation of 1, 2, 4-oxadiazole derivatives as novel GPR119 agonists

Suhong Fu1, Wei Xiang1, Jinying Chen1

  • 1State Key Laboratory of Biotherapy and Cancer Center/Collaborative Innovation Center of Biotherapy, West China Hospital, West China Medical School of Sichuan University, Chengdu, China.

Chemical Biology & Drug Design
|October 26, 2016
PubMed

Keywords:
GPCRGPR119SAR studyagonistic activitycAMP

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