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A Direct, Early Stage Guanidinylation Protocol for the Synthesis of Complex Aminoguanidine-containing Natural Products
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A Direct, Early Stage Guanidinylation Protocol for the Synthesis of Complex Aminoguanidine-containing Natural Products

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Synthesis and biological evaluation of chalcone derivatives containing aminoguanidine or acylhydrazone moieties

Zhi-Yu Wei1, Ke-Qiang Chi2, Zhan-Kui Yu1

  • 1Key Laboratory of Natural Resources and Functional Molecules of the Changbai Mountain, Affiliated Ministry of Education, Yanbian University College of Pharmacy, Yanji, Jilin Province 133002, PR China.

Bioorganic & Medicinal Chemistry Letters
|November 16, 2016
PubMed

Keywords:
AcylhydrazoneAminoguanidineAnti-inflammatory activityAntibacterial activityAntifungal activityChalconeCytotoxicity

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