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Updated: Mar 12, 2026

Continuous Fluorescence-Based Endonuclease-Coupled DNA Methylation Assay to Screen for DNA Methyltransferase Inhibitors
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Continuous Fluorescence-Based Endonuclease-Coupled DNA Methylation Assay to Screen for DNA Methyltransferase Inhibitors

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Probes and Targets of DNA Methylation and Demethylation in Drug Development

Barsam Mirfattah1, Jason Herring1, Hui Tang1

  • 1Department of Pharmacology and Toxicology, The University of Texas Medical Branch, Galveston, TX, United States.

Current Topics in Medicinal Chemistry
|November 17, 2016
PubMed

Keywords:
DNA methylationDNA methyltransferase inhibitor (DNMTi) drugscancermass spectrometry

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