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Facile Preparation of 4-Substituted Quinazoline Derivatives
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Published on: February 15, 2016

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The discovery of quinoline based single-ligand human H1 and H3 receptor antagonists

Panayiotis A Procopiou1, Rachael A Ancliff1, Paul M Gore1

  • 1Medicinal Chemistry, GlaxoSmithKline Medicines Research Centre, Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, United Kingdom.

Bioorganic & Medicinal Chemistry Letters
|November 22, 2016
PubMed

Keywords:
Allergic rhinitisH(1)H(3) histamine receptor antagonistNasal congestionQuinolineSingle ligand

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