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Developing piperlongumine-directed glutathione S-transferase inhibitors by an electrophilicity-based strategy

Hai-Bo Wang1, Xiao-Ling Jin1, Jia-Fang Zheng1

  • 1State Key Laboratory of Applied Organic Chemistry, Lanzhou University, 222 Tianshui Street S., Lanzhou, Gansu 730000, China.

European Journal of Medicinal Chemistry
|December 4, 2016
PubMed

Keywords:
ElectrophilicityGlutathione S-transferasesMultiple drug resistancePiperlongumine

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