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Synthesis and SAR evaluation of novel thioridazine derivatives active against drug-resistant tuberculosis

Nicolò Scalacci1, Alistair K Brown2, Fernando R Pavan3

  • 1Institute of Pharmaceutical Science, King's College London, 150 Stamford Street, London, SE1 9NH, United Kingdom; Northumbria University Newcastle, Department of Applied Sciences, Ellison Building, Ellison Place, NE1 8ST, Newcastle upon Tyne, United Kingdom.

European Journal of Medicinal Chemistry
|January 1, 2017
PubMed

Keywords:
Efflux pumpIndoleMDR-TBThioridazineTuberculosis

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