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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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New pyridazinone-4-carboxamides as new cannabinoid receptor type-2 inverse agonists: Synthesis, pharmacological data

Giulio Ragusa1, María Gómez-Cañas2, Paula Morales3

  • 1Department of Chemistry and Pharmacy, University of Sassari, via F. Muroni 23/A, 07100, Sassari, Italy.

European Journal of Medicinal Chemistry
|January 15, 2017
PubMed

Keywords:
ADME modelCB(2) antagonismCannabinoid receptorsDocking studiesScaffold hoppingSynthesis

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