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In Vivo Dearomatization of the Potent Antituberculosis Agent BTZ043 via Meisenheimer Complex Formation

Florian Kloss1,2, Viktor Krchnak3,4, Anna Krchnakova3

  • 1Transfer Group Antiinfectives, Leibniz Institute for Natural Product Research and Infection Biology, HKI, Beutenbergstrasse 11a, 07745, Jena, Germany.

Angewandte Chemie (International Ed. in English)
|January 19, 2017
PubMed

Keywords:
DprE1 inhibitorsbenzothiazinonesmetabolite identificationprodrugstransient metabolites

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