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Updated: Mar 8, 2026

Constructing Thioether/Vinyl Sulfide-tethered Helical Peptides Via Photo-induced Thiol-ene/yne Hydrothiolation
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Constructing Thioether/Vinyl Sulfide-tethered Helical Peptides Via Photo-induced Thiol-ene/yne Hydrothiolation

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Methanethiosulfonate derivatives as ligands of the STAT3-SH2 domain

Elena Gabriele1, Chiara Ricci2, Fiorella Meneghetti1

  • 1a Department of Pharmaceutical Sciences , Università degli Studi di Milano , Milano , Italy.

Journal of Enzyme Inhibition and Medicinal Chemistry
|January 19, 2017
PubMed

Keywords:
Anticancer drugS3I-201 analogsSH2 antagonistSTAT3cytotoxicity

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