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Updated: Mar 8, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Discovery of Chromane Propionic Acid Analogues as Selective Agonists of GPR120 with in Vivo Activity in Rodents

Gregory L Adams1, Francisco Velazquez2, Charles Jayne2

  • 1Merck & Co., Inc. , West Point, Pennsylvania 19486, United States.

ACS Medicinal Chemistry Letters
|January 21, 2017
PubMed

Keywords:
FFAR4GPR120chromaneinsulin sensitizationtype 2 diabetes

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