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Investigation of orexin-2 selective receptor antagonists: Structural modifications resulting in dual orexin receptor

Jason W Skudlarek1, Christina N DiMarco1, Kerim Babaoglu2

  • 1Department of Medicinal Chemistry, MRL, Merck & Co., Inc., West Point, PA 19486, USA.

Bioorganic & Medicinal Chemistry Letters
|February 21, 2017
PubMed

Keywords:
AntagonistGPCRInsomniaOrexinSleep

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