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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Structure-activity relationship studies of 1,7-diheteroarylhepta-1,4,6-trien-3-ones with two different terminal rings

Rubing Wang1, Xiaojie Zhang1, Chengsheng Chen1

  • 1Department of Chemistry, California State University, Fresno, 2555 E. San Ramon Avenue, M/S SB70, Fresno, CA 93740, USA.

European Journal of Medicinal Chemistry
|April 8, 2017
PubMed

Keywords:
1,7-Diheteroarylhepta-1,4,6-trien-3-oneAntiproliferative activityCell apoptosisProstate cancerStructure-activity relationship

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