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Updated: Aug 2, 2026

System for Efficacy and Cytotoxicity Screening of Inhibitors Targeting Intracellular Mycobacterium tuberculosis
09:57

System for Efficacy and Cytotoxicity Screening of Inhibitors Targeting Intracellular Mycobacterium tuberculosis

Published on: April 5, 2017

Structural analysis of the interaction between spiroisoxazoline SMARt-420 and the Mycobacterium tuberculosis

Alexandre Wohlkönig1, Han Remaut1, Martin Moune2

  • 1Center for Structural Biology, Vlaams Instituut voor Biotechnology (VIB), Pleinlaan 2, B-1050 Brussels, Belgium; Structural Biology Brussels, Vrije Universiteit Brussel (VUB), Pleinlaan 2, B-1050 Brussels, Belgium.

Biochemical and Biophysical Research Communications
|April 19, 2017
PubMed

Keywords:
Crystal structureDrug designEthionamideLigand-binding interactionTetR familyTranscriptional repressor

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