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Apparent CB1 Receptor Rimonabant Affinity Estimates: Combination with THC and Synthetic Cannabinoids in the Mouse In

T W Grim1, A J Morales2, B F Thomas2

  • 1Department of Pharmacology, Virginia Commonwealth University, Richmond, Virginia (T.W.G., A.J.M., S.S.N., A.H.L.); RTI International, Research Triangle Park, North Carolina (B.F.T., J.L.W.); and PinPoint Testing, LLC, AR (G.W.E.) tgrim@scripps.edu.

The Journal of Pharmacology and Experimental Therapeutics
|April 27, 2017
PubMed
Summary

Synthetic cannabinoids (SCs) largely exert their effects through cannabinoid 1 receptors (CB1Rs). Quantitative analysis confirmed CB1R mediation of SCs

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