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Alkyne-linked reduction-activated protecting groups for diverse functionalization on the backbone of oligonucleotides

Hisao Saneyoshi1, Kazuhiko Kondo1, Koichi Iketani1

  • 1Department of Material and Life Chemistry, Faculty of Engineering, Kanagawa University, 3-27-1 Rokkakubashi, Kanagawa-ku, Yokohama 221-8686, Japan.

Bioorganic & Medicinal Chemistry
|May 3, 2017
PubMed

Keywords:
ConjugationDrug deliveryOligonucleotide therapeuticsProtecting group

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