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A Semi-High-Throughput Adaptation of the NADH-Coupled ATPase Assay for Screening Small Molecule Inhibitors
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Insights into the myosin II inhibitory potency of A-ring-modified (S)-blebbistatin analogs

Sigrid Verhasselt1, Christian V Stevens1, Tom Van den Broecke1

  • 1SynBioC Research Group, Department of Sustainable Organic Chemistry and Technology, Campus Coupure, Ghent University, Coupure Links 653, 9000 Ghent, Belgium.

Bioorganic & Medicinal Chemistry Letters
|May 18, 2017
PubMed

Keywords:
A-ring modificationBlebbistatinMyosin II

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