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Novel delta opioid receptor agonists with oxazatricyclodecane structure showing potent agonistic activities

Kohei Hayashida1, Shigeto Hirayama2, Takashi Iwai3

  • 1Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan; Discovery Research Laboratories, Nippon Chemiphar Co., Ltd., 1-22, Hikokawado, Misato, Saitama 341-0005, Japan.

Bioorganic & Medicinal Chemistry Letters
|May 20, 2017
PubMed

Keywords:
Accessory siteDOR agonistDioxamethylene moietyOpioidOxazatricyclodecane structure

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