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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Modulation of CB1 cannabinoid receptor by allosteric ligands: Pharmacology and therapeutic opportunities

Leepakshi Khurana1, Ken Mackie2, Daniele Piomelli3

  • 1Department of Pharmaceutical Sciences, University of Connecticut, Storrs, CT 06269, United States.

Neuropharmacology
|May 22, 2017
PubMed

Keywords:
Allosteric modulatorBiased signalingCB(1)Therapeutic potential

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