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Discovery of BI 135585, an in vivo efficacious oxazinanone-based 11β hydroxysteroid dehydrogenase type 1 inhibitor

Linghang Zhuang1, Colin M Tice1, Zhenrong Xu1

  • 1Medicinal Chemistry, Vitae Pharmaceuticals, Inc, 502 West Office Center Drive, Fort Washington, PA 19034, United States.

Bioorganic & Medicinal Chemistry
|May 22, 2017
PubMed

Keywords:
11beta hydroxysteroid dehydrogenase type 1Human adipocyteHuman adipose tissueInhibitorOxazinanone

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