Voltage gated ion channels blockade is the underlying mechanism of BIMU8 induced cardiotoxicity

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Updated: Jan 24, 2026

Controllable Ion Channel Expression through Inducible Transient Transfection
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Controllable Ion Channel Expression through Inducible Transient Transfection

Published on: February 17, 2017

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Shahid Muhammad Iqbal1, Rosa Lemmens-Gruber2

  • 1Department of Pharmacology and Toxicology, University of Vienna, Althanstrasse-14 (UZA 2), A-1090 Vienna, Austria; Drug Regulatory Authority of Pakistan, Telecom Foundation (TF) Complex G-9/4, Islamabad, Pakistan.

Toxicology Letters
|May 30, 2017
PubMed

Keywords:
BIMU8Ca(V)1.2Cardiac ion channel blockadeNa(V)1.5hERG

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