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Thiophene/thiazole-benzene replacement on guanidine derivatives targeting α2-Adrenoceptors

Aoife Flood1, Cristina Trujillo1, Goar Sanchez-Sanz2

  • 1School of Chemistry, Trinity Biomedical Sciences Institute, Trinity College Dublin, 152-160 Pearse Street, Dublin 2, Ireland.

European Journal of Medicinal Chemistry
|June 24, 2017
PubMed

Keywords:
Affinity constantsAntagonistsAromaticityBioisosterismGuanidiniumThiazoleThiopheneα(2)-Adrenoceptors

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