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Discovery of highly selective κ-opioid receptor agonists: 10α-Hydroxy TRK-820 derivatives

Shinya Suzuki1, Yuji Sugawara1, Riichiro Tsuji1

  • 1Pharmaceutical Research Laboratories, Toray Industries, Inc., 6-10-1 Tebiro, Kamakura, Kanagawa 248-8555, Japan.

Bioorganic & Medicinal Chemistry Letters
|July 10, 2017
PubMed

Keywords:
4,5-EpoxymorphinanAnalgesicAntipruriticTRK-820κ-Opioid receptorμ-Opioid receptor

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