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Synthesis of novel 13α-estrone derivatives by Sonogashira coupling as potential 17β-HSD1 inhibitors

Ildikó Bacsa1, Rebeka Jójárt1, János Wölfling1

  • 1Department of Organic Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary.

Beilstein Journal of Organic Chemistry
|July 12, 2017
PubMed

Keywords:
13α-estrone17β-HSD1 inhibitionSonogashira couplingbenzofuranpartial saturation

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