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Cycloalkane analogues of sinefungin as EHMT1/2 inhibitors

Qing Liu1, Xiaoqing Cai2, Dehua Yang2

  • 1School of Pharmacy, Fudan University, Shanghai 201203, China; The CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China; The National Center for Drug Screening, Shanghai 201203, China.

Bioorganic & Medicinal Chemistry
|July 26, 2017
PubMed

Keywords:
Cycloalkyl substituted analogueMethyltransferase inhibitorNatural productSinefungin

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