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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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A computational study of the influence of methyl substituents on competitive ring closure to α- and β-lactones

Philippe B Wilson1, Ian H Williams

  • 1Leicester School of Pharmacy, De Montfort University, The Gateway, Leicester, LE1 9BH, UK.

Organic & Biomolecular Chemistry
|August 19, 2017
PubMed

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