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Discovery of novel steroidal histamine H3 receptor antagonists/inverse agonists

Istvan Ledneczki1, Pál Tapolcsányi1, Eszter Gábor1

  • 1Chemical Works of Gedeon Richter Plc, H-1475, Budapest P.O. Box 27, Hungary.

Bioorganic & Medicinal Chemistry Letters
|September 11, 2017
PubMed

Keywords:
Antagonist/inverse agonistDipsogenia modelEstrane derivativesHistamine H(3) receptorSteroid

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