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Updated: Feb 22, 2026

Regioselective O-Glycosylation of Nucleosides via the Temporary 2',3'-Diol Protection by a Boronic Ester for the Synthesis of Disaccharide Nucleosides
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Regioselective O-Glycosylation of Nucleosides via the Temporary 2',3'-Diol Protection by a Boronic Ester for the Synthesis of Disaccharide Nucleosides

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Fluorinated nucleosides as an important class of anticancer and antiviral agents

Alessandra Cavaliere1,2, Katrin C Probst2, Andrew D Westwell1

  • 1School of Pharmacy & Pharmaceutical Sciences, Cardiff University, Redwood Building, King Edward VII Avenue, Cardiff, CF10 3NB Wales, UK.

Future Medicinal Chemistry
|September 21, 2017
PubMed

Keywords:
NRTIsPET imagingRThENThuman equilibrative nucleoside transporter proteinsnucleoside analogsphosphoramidates (ProTides)reverse transcriptase

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