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Updated: Feb 21, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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Adhesion G Protein-Coupled Receptors as Drug Targets

Ryan H Purcell1, Randy A Hall1

  • 1Department of Pharmacology, Emory University School of Medicine, Atlanta, Georgia, 30322, USA;

Annual Review of Pharmacology and Toxicology
|October 3, 2017
PubMed

Keywords:
agonistantagonistantibodyligandpharmaceuticaltherapeutic

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