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Regioselective O-Glycosylation of Nucleosides via the Temporary 2',3'-Diol Protection by a Boronic Ester for the Synthesis of Disaccharide Nucleosides
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8-Mercaptoguanine Derivatives as Inhibitors of Dihydropteroate Synthase

Matthew L Dennis1,2, Michael D Lee1,2, Jitendra R Harjani1

  • 1Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, 3052, Victoria, Australia.

Chemistry (Weinheim an Der Bergstrasse, Germany)
|November 25, 2017
PubMed

Keywords:
DHPSantibioticsdrug discoveryinhibitorspterinsubstrate-envelope hypothesis

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