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Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine

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Solid-phase organic synthesis of chiral, non-racemic 1,2,4-trisubstituted 1,4-diazepanes with high σ1 receptor

Lena Fanter1, Dirk Schepmann1, Bernhard Wünsch1,2

  • 1Institut für Pharmazeutische und Medizinische Chemie, Universität Münster, Münster, Germany.

Archiv Der Pharmazie
|December 12, 2017
PubMed

Keywords:
1,2,4-trisubstituted 1,4-diazepaneschiral-pool synthesissolid-phase organic synthesissubtype selectivityσ1 receptor ligands

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