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In Vitro Imaging and Quantification of the Drug Targeting Efficiency of Fluorescently Labeled GnRH Analogues
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Recent Development of Non-Peptide GnRH Antagonists

Feng-Ling Tukun1, Dag Erlend Olberg2,3, Patrick J Riss4,5,6

  • 1School of Pharmacy, University of Oslo, 0316 Oslo, Norway. f.l.tukun@kjemi.uio.no.

Molecules (Basel, Switzerland)
|December 14, 2017
PubMed
Summary

New small molecule non-peptide antagonists offer an alternative to peptide-based gonadotropin-releasing hormone (GnRH) treatments for hormone-dependent diseases, addressing limitations of current therapies.

Keywords:
GnRH receptornon-peptide GnRH antagonist

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