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Updated: Feb 17, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Class C G protein-coupled receptors: reviving old couples with new partners

Thor C Møller1, David Moreno-Delgado1, Jean-Philippe Pin1

  • 1Institut de Génomique Fonctionnelle (IGF), CNRS, INSERM, Univ. Montpellier, 34094 Montpellier, France.

Biophysics Reports
|December 15, 2017
PubMed

Keywords:
Activation mechanismDimerizationG protein-coupled receptorsGABAGlutamate

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