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An Efficient Method for the Conjugation of Hydrophilic and Hydrophobic Components by Solid-Phase-Assisted Disulfide

Kyohei Muguruma1, Takuya Shirasaka1, Daichi Akiyama1

  • 1Department of Medicinal Chemistry, Tokyo University of Pharmacy and Life Sciences, 1432-1 Horinouchi, Hachioji, Tokyo, 192-0392, Japan.

Angewandte Chemie (International Ed. in English)
|December 26, 2017
PubMed

Keywords:
peptide-drug conjugatesolid-phase synthesissolubilitysynthetic methods

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