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A convenient transesterification method for synthesis of AT2 receptor ligands with improved stability in human liver

Johan Wannberg1, Rebecka Isaksson2, Ulf Bremberg1

  • 1Department of Medicinal Chemistry, Science for Life Laboratory, BMC, Uppsala University, P.O. Box 574, SE-751 23 Uppsala, Sweden.

Bioorganic & Medicinal Chemistry Letters
|December 28, 2017
PubMed

Keywords:
AT(2)R antagonistsAngiotensin II type 2 receptor antagonistsLiver microsomesSulfonyl carbamatesTransesterification

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