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Assaying Protein Kinase Activity with Radiolabeled ATP
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Assaying Protein Kinase Activity with Radiolabeled ATP

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Discovery of MK-8722: A Systemic, Direct Pan-Activator of AMP-Activated Protein Kinase

Danqing Feng1, Tesfaye Biftu1, F Anthony Romero1

  • 1Medicinal Chemistry, PPDM Preclinical ADME, In Vitro Pharmacology, In Vivo Pharmacology, and Biology-Discovery Departments, Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, New Jersey 07033, United States.

ACS Medicinal Chemistry Letters
|January 20, 2018
PubMed

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