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Novel aromatic sulfonyl naphthalene-based boronates as 20S proteasome inhibitors

Hongwu Liu1, Jianwei Wu1, Ying Ge1

  • 1Jiangsu Key Laboratory of Drug Design and Optimization, China Pharmaceutical University, Nanjing 210009, China.

Bioorganic & Medicinal Chemistry
|February 11, 2018
PubMed

Keywords:
20S proteasome inhibitorsBortezomibMetabolic stabilityNon-peptide scaffold

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