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O6C-20-nor-salvinorin A is a stable and potent KOR agonist

Shun Hirasawa1, Min Cho1, Tarsis F Brust2

  • 1The Scripps Research Institute, Department of Chemistry, La Jolla, CA 92037, United States.

Bioorganic & Medicinal Chemistry Letters
|February 11, 2018
PubMed

Keywords:
Conformational analysisHeck reactionKappa opioid receptorSalvinorinTotal synthesis

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