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Updated: Feb 14, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Small Molecule Allosteric Modulators of G-Protein-Coupled Receptors: Drug-Target Interactions

Shaoyong Lu1, Jian Zhang1

  • 1Department of Pathophysiology, Key Laboratory of Cell Differentiation and Apoptosis of Chinese Ministry of Education, School of Medicine , Shanghai Jiao Tong University , Shanghai 200025 , China.

Journal of Medicinal Chemistry
|February 20, 2018
PubMed

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