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High-Throughput Kinetic Analysis for Target-Directed Covalent Ligand Discovery

Gregory B Craven1,2, Dominic P Affron1, Charlotte E Allen1

  • 1Department of Chemistry, Imperial College London, South Kensington Campus, London, SW7 2AZ, UK.

Angewandte Chemie (International Ed. in English)
|February 27, 2018
PubMed

Keywords:
Cdk2covalent inhibitionfragment-based drug discoverykineticsprotein modification

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