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Updated: Feb 13, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Identification of novel agonists and antagonists of the ecdysone receptor by virtual screening

Xueping Hu1, Bin Yin1, Kaat Cappelle2

  • 1Department of Applied Chemistry, College of Science, China Agricultural University, Beijing 100193, China.

Journal of Molecular Graphics & Modelling
|March 13, 2018
PubMed

Keywords:
AgonistsAntagonistsEcdysone receptorMolecular dockingMolecular dynamic simulationVirtual screening

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