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An ELISA Based Binding and Competition Method to Rapidly Determine Ligand-receptor Interactions
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Development of novel pyridazinone-based adenosine receptor ligands

Daniela Catarzi1, Flavia Varano1, Matteo Falsini1

  • 1Dipartimento di Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino, Sezione di Farmaceutica e Nutraceutica, Università degli Studi di Firenze, Via Ugo Schiff, 6, 50019 Sesto Fiorentino, Italy.

Bioorganic & Medicinal Chemistry Letters
|April 9, 2018
PubMed

Keywords:
ADME propertiesAdenosine receptor ligandsG protein-coupled receptorsThieno[2,3-d]pyridazin-5(4H)-ones

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