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Reversible, orally available ADP receptor (P2Y12) antagonists Part I: Hit to lead process

Imadul Islam1, Shendong Yuan2, Robert G Wei2

  • 1Medical Core Facility and Research Platforms, King Abdullah International Medical Research Center/King Saud bin Abdulaziz University for Health Sciences, Ministry of National Guard-Health Affairs, Riyadh 11426, Saudi Arabia; Department of Medicinal Chemistry, Berlex Biosciences, 2600 Hilltop Drive, Richmond, CA 94804, United States.

Bioorganic & Medicinal Chemistry Letters
|April 10, 2018
PubMed

Keywords:
ADPAntiplatelet therapyHTSP2Y(12) antagonistsParallel synthesis

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